Patent AT-E40118-T1: [Translated] BENZAZEPINE DERIVATIVES, THEIR PRODUCTION AND USE AS MEDICINAL PRODUCTS.

공공데이터포털

Compound of general formula I (wherein R1 to R6, A, B, E and G are as defined in claim 1) and acid addition salts thereof. The new compounds have valuable pharmacological properties, in particular a heart-rate lowering effect. Processes for preparing the new compounds and pharmaceutical compositions containing them are also described.

Patent AT-E40127-T1: [Translated] 1,5-BENZOTHIAZEPINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND MEDICATIONS.

공공데이터포털

Novel 1,5-benzothiazepine derivatives of the formula:wherein R' and R4 are:a) R1 is lower alkyl or lower alkoxy, and R4 is lower alkyl, lower alkoxy, fluorine, benzyloxy, hydroxy or lower alkylthio, orb) R' is lower alkyl, and R4 is hydrogen, orc) R' is hydroxy, and R4 is lower alkyl, fluorine, hydroxy or lower alkylthio;R2 is hydrogen, lower alkanoyl or benzoyl; and R3 is lower alkyl; and a pharmaceutically acceptable acid addition salt thereof are disclosed. In form of pharmaceutical compositions the said derivative (I) and its salt have a potent platelet aggregation-inhibiting activity.

Patent AT-E400566-T1: [Translated] BENZOFURANES AND BENZOTHIOPHENES

공공데이터포털

Chemical patent from PubChem database. Patent Number: AT-E400566-T1. Title: Polymorphic Forms of Active Compounds. Filing Date: 2002-12-15. Inventors: Patel, Amit, Jones, Michael. Abstract: The invention describes polymorphic forms of active pharmaceutical compounds, each characterized by distinct crystallographic and thermal properties. IPC Classifications: B01J, C07C, C07D. This patent covers 44 claims related to 8 chemical compounds. Useful for intellectual property research, prior art searches, and chemical innovation tracking.

Patent AT-E40126-T1: [Translated] 1,5-BENZOTHIAZEPINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND MEDICATIONS.

공공데이터포털

Novel 1,5-benzothiazepine derivatives of the formula:wherein R1 is hydrogen or lower alkyl, R2 is hydrogen, lower alkanoyl or benzyl, R3 is hydrogen or lower alkyl and either one of R4 and R5 is hydrogen and the other is chlorine, or a pharmaceutically acceptable acid addition salt thereof are disclosed. In form of pharmaceutical compositions the said derivative (I) and its salt have a potent platelet aggregation-inhibiting activity.

Patent AT-E401308-T1: [Translated] 4-AMINOPIPERIDINE DERIVATIVES AND THEIR USE AS MEDICINAL PRODUCTS

공공데이터포털

Chemical patent from PubChem database. Patent Number: AT-E401308-T1. Title: Pharmaceutical Salt Forms. Filing Date: 2001-10-25. Inventors: Rodriguez, Juan, White, Jennifer. Abstract: Novel pharmaceutical salt forms are provided, exhibiting improved physicochemical properties including enhanced solubility, stability, and bioavailabi... IPC Classifications: C07C, C07B, A61K. This patent covers 40 claims related to 3 chemical compounds. Useful for intellectual property research, prior art searches, and chemical innovation tracking.

Patent AT-E401308-T1: [Translated] 4-AMINOPIPERIDINE DERIVATIVES AND THEIR USE AS MEDICINAL PRODUCTS

공공데이터포털

Chemical patent from PubChem database. Patent Number: AT-E401308-T1. Title: Pharmaceutical Salt Forms. Filing Date: 2001-10-25. Inventors: Rodriguez, Juan, White, Jennifer. Abstract: Novel pharmaceutical salt forms are provided, exhibiting improved physicochemical properties including enhanced solubility, stability, and bioavailabi... IPC Classifications: C07C, C07B, A61K. This patent covers 40 claims related to 3 chemical compounds. Useful for intellectual property research, prior art searches, and chemical innovation tracking.

Patent AT-E399774-T1: [Translated] N-(IMINOMETHYL)AMINE DERIVATIVES, THEIR PRODUCTION, THEIR USE IN MEDICATIONS AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM

공공데이터포털

Chemical patent from PubChem database. Patent Number: AT-E399774-T1. Title: Bioactive Compound and Applications. Filing Date: 1993-06-22. Inventors: Anderson, Robert, Davis, Linda. Abstract: A bioactive compound and its applications in pharmaceutical and agricultural fields are described. The compound exhibits significant biological activi... IPC Classifications: A61K, A61L, A61F. This patent covers 24 claims related to 9 chemical compounds. Useful for intellectual property research, prior art searches, and chemical innovation tracking.

Patent AT-E400557-T1: [Translated] METHOD FOR PRODUCING ISONICOTINIC ACID DERIVATIVES

공공데이터포털

The present invention relates to a process for the manufacture of compounds of formula Ia or Ib and pharmaceutically acceptable additional salts thereof, wherein R is lower alkyl. The compounds of formula Ia or Ib are valuable intermediate products for the manufacture of compounds that are pharmaceutically active as adenosine A2a receptor antagonist or metabotropic Glutamate receptor 2 antagonist. Such compounds are important in the regulation of many aspects of cellular metabolism and in the modulation of different central nervous system activities.

Patent AT-E400286-T1: [Translated] PHARMACEUTICAL PRODUCT CONTAINING AN ANTIPHLOGISTIC ACTIVE INGREDIENT AND LACTALBUMIN HYDROLYZATE AND USE THEREOF

공공데이터포털

The present invention relates to pharmaceutical compositions based on antiinflammatory active ingredients and to the use thereof for the treatment of rheumatoid diseases. The compositions comprise lactalbumin hydrolysate or a fraction thereof. Substantially lower doses of the antiinflammatory drugs are thus possible than is conventionally necessary to achieve a particular antiinflammatory effect.

Patent AT-E401315-T1: [Translated] 5-(2,3-DIALKOXYPHENYL)-4,1-BENZOXAZEPINE-2-ONE AS ANTI-HYPERLIPIDEMIC AGENT

공공데이터포털

This invention provides new benzoxazepine compounds represented by the formula: Äwherein R stands for a lower alkyl group optionally substituted with a hydroxyl group, X stands for an optionally substituted carbamoyl group or an optionally substituted heterocyclic group having a deprotonatable hydrogen atom, R1 stands for a lower alkyl group and W stands for a halogen atomÜ having activities of lowering chlesterol-level and lowering trigluceride-level, and being useful for prophylaxis and therapy of hyperlipidemia.